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Olmesartan Medoxomil is an angiotensin receptor blocker (ARB) that lowers blood pressure and prevents heart problems. Find out more about its uses, side effects, drug interactions and available medicines on 1mg.com, India's largest healthcare platform. Olmesartan Medoxomil is a medication that lowers blood pressure by blocking angiotensin II receptors. It can also help diabetic patients prevent kidney damage and is available in 20 mg and 40 mg doses. Olmesartan medoxomil, a prodrug, is hydrolyzed to olmesartan during absorption from the gastrointestinal tract. Olmesartan is a selective AT 1 subtype angiotensin II receptor antagonist. Olmesartan is an angiotensin II receptor blocker (sometimes called an ARB). Olmesartan is used to treat high blood pressure (hypertension) in adults and children at least 6 years old.